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Cationic Liposomes Carrying siRNA: Impact of Lipid Composition on Physicochemical Properties, Cytotoxicity and Endosomal Escape
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Analysis of Genes Associated With Monogenic Primary Immunodeficiency Identifies Rare Variants in XIAP in Patients With Crohn's Disease.
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Cationic Liposomes Carrying siRNA: Impact of Lipid Composition on Physicochemical Properties, Cytotoxicity and Endosomal Escape
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2018 • In Nanomaterials, 8 (5)
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Tumor cells may circulate in medullary thyroid cancer patients independently of serum calcitonin
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2018 • In Biochemical Pharmacology
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2017 • In British Journal of Pharmacology, 174 (Suppl 1), p. 1-S16
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Gallo, Robert; Willems, Luc ; Tagaya, Yutaka
2017 • In Frontiers in Microbiology, 8, p. 1800
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Metabolic inhibitors accentuate the anti-tumoral effect of HDAC5 inhibition
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2017 • In Oncogene
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Chemokine neutralization as an innovative therapeutic strategy for atopic dermatitis
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PEGylated and Functionalized Aliphatic Polycarbonate Polyplex Nanoparticles for Intravenous Administration of HDAC5 siRNA in Cancer Therapy
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2017 • In Scientific Reports, 7 (1)
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2017 • In Kidney International
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2016 • In Oncotarget
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2016 • In Pharmacology and Therapeutics
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Guidelines for the use and interpretation of assays for monitoring autophagy (3rd edition).
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Specific expression and function of inositol 1,4,5-trisphosphate 3-kinase C (ITPKC) in wild type and knock-out mice
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EGFR tyrosine kinase inhibitors overcome resistance to chemotherapy in malignant pleural mesothelioma.
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2016 • In Proceedings of the 107th Annual Meeting of the American Association for Cancer Research; 2016 Apr 16-20; New Orleans, LA. Philadelphia (PA): AACR; Cancer Res 2016
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2015 • In ERJ Open Research, 1 (2)
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2015 • In ERJ Open Research, 1 (2), p. 00028
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2015 • In Viruses, 7, p. 3603-3624
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Willems, Luc ; Gillet, Nicolas
2015 • In Viruses, 7, p. 2999-3018
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A fungal biofilm reactor based on metal structured packing improves the quality of a Gla::GFP fusion protein produced by Aspergillus oryzae
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Mutation of a Single Envelope N-linked Glycosylation Site Enhances the Pathogenicity of Bovine Leukemia Virus
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2015 • In BMC Cancer, 15, p. 227
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2015 • In Developmental Cell, 34, p. 400-409
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2015 • In British Journal of Haematology, 168 (2), p. 230-8
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The Ras/Rap GTPase activating protein RASA3 : from gene structure to in vivo functions
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2015 • In Advances in Biological Regulation, 57, p. 153-161
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Comparative Interactome of HIV-1 Tat and Human T Lymphotropic Virus Type-1 Tax and the Cellular Transcriptional Machinery.
Vandermeulen, Charlotte ; Hajingabo, Leon-Juvenal; Twizere, Jean-Claude
2015 • In AIDS Research and Human Retroviruses, 31 (12), p. 1204-5
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Inhiber HDAC5 : un outil pour couper court à l’immortalité des cellules cancéreuses
Polese, Catherine ; Mottet, Denis
2014 • In MS. Medecine Sciences, 30 (numero 8-9), p. 730-732
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Rates of CTL Killing in Persistent Viral Infection In Vivo
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2014 • In PLoS Computational Biology, 4
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2014 • In Bioprocess and Biosystems Engineering
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2014 • In Vascular Pharmacology, 60, p. 57-66
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The Tax protein and the minichromosome maintenance protein complex MCM2-7 affect cell replication and viral transcription
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2014 • In Retrovirology, 11, p. 101
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2014 • In Retrovirology, 11 (S1), p. 90
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Hyper-replicative bovine leukemia virus by mutation of an envelope N-linked glycosylation site
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2014 • In Retrovirology, 11 (1), p. 141
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Vaccination against delta-Retroviruses: The Bovine Leukemia Virus Paradigm.
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2014 • In Viruses, 6 (6), p. 2416-2427
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Predicting interactome networks perturbations in human cancer: application to gene fusions in acute lymphoblastic leukemia.
Juvenal Hajingabo, Leon; Daakour, Sarah ; Martin, Maud et al.
2014 • In Molecular Biology of the Cell
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An Easy, Convenient Cell and Tissue Extraction Protocol for Nuclear Magnetic Resonance Metabolomics.
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2014 • In Phytochemical Analysis, 25, p. 342-349
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Rasa3 Controls Megakaryocyte Rap1 Activation, Integrin Signaling and Differentiation into Proplatelet
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2014 • In PLoS Genetics, 10 (6), p. 1004420
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DNA Damage and Thyroid Cancer
Neelature Sriramareddy, Sathyanarayana ; Staumont, Bernard ; Willems, Luc
2014 • In GIGADay-2014
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Generation and validation of a mouse model for conditional inactivation of PLAGL1
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2014 • In Proceedings of the 4th edition : FARAH Day 2014
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A proteome-scale map of the human interactome network.
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2014 • In Cell, 159 (5), p. 1212-26
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Novel activating mutations lacking cysteine in type I cytokine receptors in acute lymphoblastic leukemia.
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Inositol trisphosphate 3-kinase B is increased in human Alzheimer brain and exacerbates mouse Alzheimer pathology
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The Anti-Tumor Effect of HDAC Inhibition in a Human Pancreas Cancer Model Is Significantly Improved by the Simultaneous Inhibition of Cyclooxygenase 2
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2013 • In PLoS ONE, 8 (9), p. 75102
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A new role for histone deacetylase 5 in the maintenance of long telomeres.
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2013 • In FASEB Journal, 27
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Synthesis and pharmacological evaluation of 2-aryloxy/arylamino-5-cyanobenzenesulfonylureas as novel thromboxane A2 receptor antagonists
2013 • In European Journal of Medicinal Chemistry, 65, p. 32-40
Communication publiée dans un périodique (Colloques et congrès scientifiques)
Biophysical characterization of the interaction of novel aromatic glycolipid surfactants with membrane models.
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2013 • In World Academy of Science, Engineering and Technology, 77, p. 840
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Biophysical characterization of the interaction of novel aromatic glycolipid surfactants with membrane models.
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2013 • In World Academy of Science, Engineering and Technology, 77, p. 840
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An eYFP Reporter Gene for the Yeast Two-hybrid System
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2013 • In Protein Journal, 32 (2), p. 126-130
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The role of TGFalpha in the resistance to mesothelioma chemotherapy
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2013 • In GIGA-Day 2013
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Identification of microRNA-based signatures for response and survival for non-small cell lung cancer treated with cisplatin-vinorelbine A ELCWP prospective study
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2013 • In Lung Cancer, 82, p. 340-345
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The homeodomain transcription factor Hoxa2 interacts with and promotes the proteasomal degradation of the E3 ubiquitin protein ligase RCHY1.
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2013 • In PLoS ONE, 8 (11), p. 80387
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Direct and indirect use of GFP whole cell biosensors for the assessment of bioprocess performances: design of milliliter scale-down bioreactors
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2013 • In Biotechnology Progress, 29 (1), p. 48-59
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Thyroid-specific inactivation of Kif3a alters TSH signaling pathway and leads to hypothyroidism.
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2013 • In Journal of Molecular Endocrinology, 50, p. 375-387
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Massive Depletion of Bovine Leukemia Virus Proviral Clones Located in Genomic Transcriptionally Active Sites During Primary Infection
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2013 • In PLoS Pathogens, 9 (10)
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Heterologously expressed formyl peptide receptor 2 (FPR2/ALX) does not respond to lipoxin A4
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PP2A regulatory subunit Balpha controls endothelial contractility and vessel lumen integrity via regulation of HDAC7.
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2013 • In EMBO Journal
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Inositol 1,4,5-trisphosphate 3-kinase B (Itpkb) controls survival, proliferation and cytokine production in mouse peripheral T cells
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The role of epigenetics in malignant pleural mesothelioma
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WIP1 deficiency inhibits HTLV-1 Tax oncogenesis: novel therapeutic prospects for treatment of ATL?
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2012 • In Retrovirology, 9 (1), p. 115
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Chemoresistance to Valproate Treatment of Bovine Leukemia Virus-Infected Sheep; Identification of Improved HDAC Inhibitors
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2012 • In Pathogens, (2012-1), p. 65-82
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Interactomic map of the Ets factors family : Identification of unexpected functions in mRNA processing
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Potentiality of using microbial biosensors for the detection of substrate heterogeneities and the assessment of microbial viability in industrial bioreactors: a complete set of experiments in chemostat and scale-down reactors, and elaboration of a mini scale-down platform
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2012 • In Communications in Agricultural and Applied Biological Sciences, 77 (1), p. 3-7
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2012 • In Genes and Genomics, 34, p. 107-110
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Interaction network of antimicrobial peptides of Arabidopsis thaliana, based on hith-throughput yeast two-hybrid screening
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2012 • In Plant Physiology and Biochemistry, p. 245-252
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Developmental defects and rescue from glucose intolerance of a catalytically-inactive novel Ship2 mutant mouse
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2012 • In Cellular Signalling, 24, p. 1971-1980
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Viral expression directs the fate of B cells in BLV-infected sheep.
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2012 • In Journal of Virology, 86 (1), p. 621-624
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Hanson, Julien ; Gille, Andreas; Offermanns, Stefan
2012 • In Pharmacology and Therapeutics
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Proinflammatory Cytokines Induce Bronchial Hyperplasia and Squamous Metaplasia in Smokers: Implications for chronic obstructive pulmonary disease therapy.
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2012 • In American Journal of Respiratory Cell and Molecular Biology, 47 (1), p. 67-79
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2012 • In EMBO Journal
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2012 • In BMC Developmental Biology, 12, p. 29
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The c-jun N-terminal Kinase (JNK)-binding Protein (JNKBP1) Acts as a Negative Regulator of NOD2 Protein Signaling by Inhibiting Its Oligomerization Process
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2012 • In Journal of Biological Chemistry, 287 (35), p. 29213-26
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2012 • In Cell Death and Differentiation
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Phosphorylation of p65(RelA) on Ser547 by ATM represses NF-κB-dependent transcription of specific genes after genotoxic stress.
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2012 • In PLoS ONE
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Host-pathogen interactome mapping for HTLV-1 and -2 retroviruses.
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2012 • In Retrovirology, 9, p. 26
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The angiogenesis suppressor gene AKAP12 is under the epigenetic control of HDAC7 in endothelial cells.
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2012 • In Angiogenesis
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Transformation by deltaretroviruses: mechanisms and therapies
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2012 • In Proceedings of the Belgian Royal Academies of Medicine, 1, p. 157-165
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Safety of long-term treatment of HAM/TSP patients with valproic acid
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2011 • In Blood, 118 (9), p. 2483-2491
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Cherdon, Céline ; Rolin, Stéphanie; Hanson, Julien et al.
2011 • In Congress of the International Society of Thrombosis and Hemostasis- 57th Annual SSC Meeting
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Histone Deacetylase 7 Regulates Cell Survival and TCR Signaling in CD4/CD8 Double-Positive Thymocytes.
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2011 • In Journal of Immunology, 186 (8), p. 4782-93
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BM-573 inhibits the development of early atherosclerotic lesions in Apo E deficient mice by blocking TP receptors and thromboxane synthase.
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2011 • In Prostaglandins and Other Lipid Mediators
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NF-kappaB inhibition improves the sensitivity of human glioblastoma cells to 5-aminolevulinic acid-based photodynamic therapy.
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2011 • In Biochemical Pharmacology
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The varicella-zoster virus ORF47 kinase interferes with host innate immune response by inhibiting the activation of IRF3.
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2011 • In PLoS ONE, 9 (2)
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Identification of a Brucella spp. secreted effector specifically interacting with human small GTPase Rab2.
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2011 • In Cellular Microbiology, 13 (7), p. 1044-58
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2011 • In Biotechnology Journal, 6, p. 968-978
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2011 • In Oncogene
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Heterozygous inactivation of the Na/Ca exchanger increases glucose-induced insulin release, β-cell proliferation, and mass.
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2011 • In Diabetes, 60, p. 2076-2085
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The inositol Inpp5k 5-phosphatase affects osmoregulation through the vasopressin-aquaporin 2 pathway in the collecting system.
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Dentin Matrix Protein 1 induces membrane expression of VE-cadherin on endothelial cells and inhibits VEGF-induced angiogenesis by blocking VEGFR-2 phosphorylation.
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Valproate–doxorubicin: promising therapy for progressing mesothelioma. A phase II study
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Regulation of B cell survival, development and function by inositol 1,4,5-trisphosphate 3-kinase B (Itpkb)
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Histone deacetylases: anti-angiogenic targets in cancer therapy.
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2010 • In Current Cancer Drug Targets, 10 (8), p. 898-913
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2010 • In British Journal of Haematology, 151
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2010 • In Inserm Workshop: Interactomics: at the crossroads of biology and bioinformatics
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An autocrine lactate loop mediates insulin-dependent inhibition of lipolysis through GPR81.
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Nicotinic acid- and monomethyl fumarate-induced flushing involves GPR109A expressed by keratinocytes and COX-2-dependent prostanoid formation in mice.
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Long-term treatment with valproic acid does not alleviate the condition of HAM/TSP
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Mutations in the inositol polyphosphate-5-phosphatase E gene link phosphatidyl inositol signaling to the ciliopathies
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Reduced levels of reactive oxygen species correlate with inhibition of apoptosis, rise in thioredoxin expression and increased bovine leukemia virus proviral loads.
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2009 • In British Journal of Cancer, 101 (9), p. 1497-501
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Neuronal injury in NCX3 knockout mice following permanent focal cerebral ischemia and in NCX3 knockout cortical neuronal cultures following oxygen-glucose deprivation and glutamate exposure
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2009 • In Nature Genetics, 41, p. 1027-1031
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Gene activation therapy: from the BLV model to HAM/TSP patients.
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HDAC4 represses p21(WAF1/Cip1) expression in human cancer cells through a Sp1-dependent, p53-independent mechanism.
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Valproate, in combination with pemetrexed and cisplatin, provides additional efficacy to the treatment of malignant mesothelioma.
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The 14th International Conference on Human Retrovirology: HTLV and related retroviruses (July 1-4, 2009; Salvador, Brazil).
Willems, Luc
2009 • In Retrovirology, 6, p. 77
Article (Périodiques scientifiques)
Protein Phosphatase 2a Controls The Activity Of Histone Deacetylase 7 During T Cell Apoptosis And Angiogenesis
Martin, Maud ; Potente, M.; Janssens, V. et al.
2008 • In Proceedings of the National Academy of Sciences of the United States of America, 105 (12), p. 4727-4732
Article (Périodiques scientifiques)
How HTLV-1 may subvert miRNAs for persistence and transformation.
Bouzar, Amel ; Willems, Luc
2008 • In Retrovirology, 5, p. 101
Article (Périodiques scientifiques)
The HTLV-1 Tax interactome.
Boxus, Mathieu ; Twizere, Jean-Claude ; Legros, Sebastien et al.
2008 • In Retrovirology, 5, p. 76
Article (Périodiques scientifiques)
Reduction of B cell turnover in chronic lymphocytic leukaemia.
Defoiche, Julien; Debacq, Christophe; Asquith, Becca et al.
2008 • In British Journal of Haematology, 143 (2), p. 240-7
Article (Périodiques scientifiques)
Emphasis on cell turnover in two hosts infected by bovine leukemia virus: a rationale for host susceptibility to disease.
Florins, Arnaud-Francois ; Boxus, Mathieu ; Vandermeers, Fabian et al.
2008 • In Veterinary Immunology and Immunopathology, 125 (1-2), p. 1-7
Article (Périodiques scientifiques)
NCX3 knockout mice exhibit increased hippocampal CA1 and CA2 neuronal damage compared to wild-type mice following global cerebral ischemia
Jeffs, G. J.; Meloni, B.; Sokolow, S. et al.
2008 • In Experimental Neurology, 210, p. 268-273
Article (Périodiques scientifiques)
Inositol trisphosphate 3-kinase B (InsP3KB) as a physiological modulator of myelopoiesis
Jia, Y.; Loison, F.; Erneux, C. et al.
2008 • In Proceedings of the National Academy of Sciences of the United States of America, 105, p. 4739-4744
Article (Périodiques scientifiques)
Regulation of innate immunity by inositol 1,3,4,5-tetrakisphosphate
Jia, Y.; Schurmans, Stéphane ; Luo, H. R.
2008 • In Cell Cycle, 7, p. 2803-2808
Article (Périodiques scientifiques)
Targeted disruption of Na+/Ca2+ exchanger 3 (NCX3) gene leads to a worsening of ischemic brain damage
Molinaro, P.; Cuomo, O.; Pignataro, G. et al.
2008 • In Journal of Neuroscience, 28, p. 1179-1184
Article (Périodiques scientifiques)
Les histones desacetylases : nouvelles cibles pour les therapies anti-cancereuses.
Mottet, Denis ; Castronovo, Vincenzo
2008 • In MS. Medecine Sciences, 24 (8-9), p. 742-6
Article (Périodiques scientifiques)
Early and transient reverse transcription during primary deltaretroviral infection of sheep.
Pomier, Carole; Alcaraz, Maria Teresa Sanchez; Debacq, Christophe et al.
2008 • In Retrovirology, 5, p. 16
Article (Périodiques scientifiques)
Nucleolin binds specifically to an AP-1 DNA sequence and represses AP1-dependent transactivation of the matrix metalloproteinase-13 gene.
Samuel, Shaija; Twizere, Jean-Claude ; Beifuss, Katherine K et al.
2008 • In Molecular Carcinogenesis, 47 (1), p. 34-46
Article (Périodiques scientifiques)
Implication des modifications épigénétiques dans les cancers : développement de nouvelles approches thérapeutiques
Vandermeers, Fabian ; Kettmann, Richard ; Willems, Luc
2008 • In Biotechnologie, Agronomie, Société et Environnement, 12 (2)
Article (Périodiques scientifiques)
Newly identified biologically active and proteolysis-resistant VEGF-A isoform VEGF111 is induced by genotoxic agents
Mineur, Pierre ; Colige, Alain ; Deroanne, Christophe et al.
2007 • In Journal of Cell Biology, 179 (6), p. 1261-1273
Article (Périodiques scientifiques)
Histone deacetylase 7 silencing alters endothelial cell migration, a key step in angiogenesis
Mottet, Denis ; Bellahcene, Akeila ; Pirotte, Sophie et al.
2007 • In Circulation Research, 101 (12), p. 1237-1246
Article (Périodiques scientifiques)
Histone Deacetylases: Target Enzymes for Cancer Therapy
Mottet, Denis ; Castronovo, Vincenzo
2007 • In Clinical and Experimental Metastasis
Article (Périodiques scientifiques)
Phosphoinositide phosphatases in a network of signaling reactions
Blero, D.; Payrastre, B.; Schurmans, Stéphane et al.
2007 • In Pflügers Archiv: European Journal of Physiology, 455, p. 31-44
Article (Périodiques scientifiques)
Les chémokines et leurs récepteurs : rôle dans les infections virales et dans les pathologies cancéreuses
Burteau, C.; Willems, Luc ; Kettmann, Richard
2007 • In Biotechnologie, Agronomie, Société et Environnement
Communication publiée dans un périodique (Colloques et congrès scientifiques)
BM-573, a thromboxane receptor antagonist, reduces development of atherosclerosis in apoE–deficient mice
Cherdon, Céline ; Rolin, Stéphanie; Hanson, Julien et al.
2007 • In Journal of Molecular and Cellular Cardiology, 42 (suppl 1.), p. 33-34
Article (Périodiques scientifiques)
Cell dynamics and immune response to BLV infection: a unifying model
Florins, Arnaud-Francois ; Gillet, Nicolas ; Asquith, Becca et al.
2007 • In Frontiers in Bioscience: A Journal and Virtual Library, 12, p. 1520-1531
Article (Périodiques scientifiques)
Even attenuated bovine leukemia virus proviruses can be pathogenic in sheep.
Florins, Arnaud-Francois ; Gillet, Nicolas ; Boxus, Mathieu et al.
2007 • In Journal of Virology, 81 (18), p. 10195-200